2007 to present

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• Utilization of the Suzuki Coupling to Enhance the Antituberculosis Activity of Aryloxazoles. Moraski, G. C.; Franzblau, S. C.; Miller, M. J. Heterocycles, 2010, 80, 977-988.

• Synthesis of Dideoxymycobactin Antigens Presented by CD1a Reveals T Cell Fine Specificity for Natural Lipopeptide Structures. Young, D. C.; Kasmar, A.; Moraski, G.; et al. J. Biol. Chem, 2009, 284, 25087-25096.

• Miller, M. J.; Li, H.; Foss, C. A. "Novel antisense oligonucleotides containing hydroxamate linkages:  targeted iron-triggered chemical nucleases." Biometals, 2009, 22, 491-510.  DOI 10.1007/s10534-009-9206-7.

• Wencewicz, T. A.; Möllmann, U.; Long, T. E.; Miller, M. J. “Is drug release necessary for antimicrobial activity of siderophore-drug conjugates?  Syntheses and biological studies of the naturally occurring salmycin “Trojan Horse” antibiotics and synthetic desferridanoxamine-antibiotic conjugates.” Biometals, 2009, 22, 633-648.  DOI 10.1007/s10534-009-9218-3.

• Synthesis and Anticancer Activity of New Hydroxamic Acid Containing 1,4-Benzodiazepines. Tardibono, Lawrence P.; Miller, Marvin J.    Org. Lett.  2009,  11,  1575–1578. DOI: 10.1021/ol900210h

• Pd(0)/InI-Mediated Allylic Additions to 4-Acetoxy-2-azetidinone: New Route to Highly Functionalized Carbocyclic Scaffolds. Cesario, Cara; Miller, Marvin J. Org. Lett. 2009,  11,  1293–1295. DOI: 10.1021/ol9000685

• Syntheses of New Spirocarbocyclic Nucleoside Analogs Using Iminonitroso Diels-Alder Reactions.    Lin, Weimin; Gupta, Anuradha; Kim, Kyung Hee; Mendel, David; Miller, Marvin J. Org. Lett.  2009, 11,  449–452. DOI: 10.1021/ol802553g

• Utilization of microbial iron assimilation processes for the development of new antibiotics and inspiration for the design of new anticancer agents.    Miller, Marvin J.; Zhu, Helen; Xu, Yanping; Wu, Chunrui; Walz, Andrew J.; Vergne, Anne; Roosenberg, John M.; Moraski, Garrett; Minnick, Albert A.; McKee-Dolence, Julia; Hu, Jingdan; Fennell, Kelley; Dolence, E. Kurt; Dong, Li; Franzblau, Scott; Malouin, Francois; Mollmann, Ute. BioMetals  2009,  22,  61–75.

• Bronsted acid-mediated opening of nitroso cycloadducts under anhydrous conditions.    Bodnar, Brian S.; Miller, Marvin J. Tetrahedron Lett.  2009, 50,  796–798.

• Evolution of Natural Product Scaffolds by Acyl- and Arylnitroso Hetero-Diels-Alder Reactions: New Chemistry on Piperine. Krchnak, Viktor; Waring, Katherine R.; Noll, Bruce C.; Moellmann, Ute; Dahse, Hans-Martin; Miller, Marvin J.  J. Org. Chem. 2008, 73,  4559–4567. DOI: 10.1021/jo8004827

• Fennell, Kelley A.; Moellmann, Ute; Miller, Marvin J. Syntheses and Biological Activity of Amamistatin B and Analogs.    J. Org. Chem. 2008, 73, 1018–1024. DOI: 10.1021/jo7020532

• Solid-Supported Nitroso Hetero-Diels–Alder Reactions. 3. Acid-Mediated Transformation of Cycloadducts by Scission of the Oxazine C−O Bonds. Krchnak, Viktor; Moellmann, Ute; Dahse, Hans-Martin; Miller, Marvin J. J. Comb. Chem. 2008, 10, 112–117. DOI: 10.1021/cc700142d

• Solid-Supported Nitroso Hetero Diels–Alder Reactions. 2. Arylnitroso Dienophiles: Scope and Limitations. Krchnak, Viktor; Moellmann, Ute; Dahse, Hans-Martin; Miller, Marvin J. J. Comb. Chem. 2008, 10, 104–111. DOI: 10.1021/cc7001414

• Solid-Supported Nitroso Hetero Diels–Alder Reactions. 1. Acylnitroso Dienophiles: Scope and Limitations. Krchnak, Viktor; Moellmann, Ute; Dahse, Hans-Martin;  Miller, Marvin J. J. Comb. Chem. 2008, 10, 94–103. DOI: 10.1021/cc700140h

• Peptides selected for the protein nanocage pores change rates of iron recovery from the ferritin mineral. Liu, X. S.; Patterson, L. D.; Miller, M. J.; Theil, E. C. J. Biol. Chem. 2007, 282, 31821–31825.DOI: 10.1074/jbc.C700153200

• Iminonitroso Diels-Alder Reactions for Efficient Derivatization and Functionalization of Complex Diene-Containing Natural Products. Li, F.; Yang, B.; Miller, M. J.; Zajicek, J.; Noll, B. C.; Möllmann, U.; Dahse, H.-M.; Miller, P. A. Org. Lett. 2007, 9, 2923-2926. DOI: 10.1021/ol071322b
  

• ß-Lactams in Synthesis: Short Syntheses of Cobactin Analogs. Walz, A. J.; Miller, M. J. Tetrahedron Letters 2007, 48, 5103-5105. DOI: 10.1016/j.tetlet.2007.05.085
  

• Synthesis and Studies of Catechol-Containing Mycobactin S and T Analogs. Walz, A. J.; Möllmann, U. Org. Biomol. Chem. 2007, 5, 1621-1628. DOI: 10.1039/b703116e
  

• Syntheses of Amamistatin Fragments and Determination of their HDAC and Antitumor Activity. Fennell, K. A.; Miller, M. J. Org. Lett., 2007, 9, 1683-1685. DOI: 10.1021/ol070382e
  

• Reactions of Nitroso Hetero Diels-Alder Cycloadducts with Azides: Stereoselective Formation of Triazolines and Aziridines. Bodnar, B. S.; Miller, M. J. J. Org. Chem., 2007, 79, 3929-3932. DOI: 10.1021/jo0701987
  

• Synthesis and biological activity of saccharide based lipophilic siderophore mimetics as potential growth promoters for mycobacteria. Gebhardt, P.; Crumbliss, A. L.; Miller, M. J.; Möllmann, U. Biometals 2007, in press. DOI: 10.1007/s10534-007-9091-x

• Syntheses and Anti-HIV Activities of (±)-Norcarbovir and (±)-Norabacavir. Huang, W.; Miller, M. J.; De Clercq, E.; Balzarini, J. Org. Biomol. Chem., 2007, 5, 1164-1166. DOI: 10.1039/b700321h
  

• Design, synthesis and pharmacological activity of novel enantiomercially pure phosphonic acid-based NAALADase inhibitors. Ding, P.; Helquist, P.; Miller, M. J. Org. Biomol. Chem. 2007, 5, 826-831. DOI: 10.1039/b615603g
  

• Azetidinones as vasopressin Via antagonists. Guillon, C. D.; Koppel, G. A.; Brownstein, M. J.; Chaney, M. O.; Ferris, C. F.; Lu, S.-F.; Fabio, K. M.; Miller, M. J.; Heindel, N. D.; Hunden, D. C.; Cooper, R. D. G.; Kaldor, S. W.; Skelton, J. J.; Dressman, B. A.; Clay, M. P.; Steinberg, M. I.; Bruns, R. F.; Simon, N. G. Bioorg. Med. Chem. 2007, 15, 2054-2080. DOI: 10.1016/j.bmc.2006.12.031
  

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2000-2006

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• Orally active vasopressin V1a receptor antagonist, SRX251, selectively blocks aggressive behavior. Ferris, C. F.; Lu, S.-F.; Messenger, T.; Guillon, C. D.; Heindel, N.; Miller, M.; Koppel, G.; Bruns, R. F.; Simon, N. G. Pharmacol. Biochem. and Behav.2006, 83, 169-174. DOI: 10.1016/j.pbb.2006.01.001
• New C-3' Hydroxamate-substituted and More Lipophilic Cyclic Hydroxamate Cephalosporin Derivatives as a Potential New Generation of Selective Antimicrobial Agents. Miller, M. J.; Zhao, G.; Vakulenko, S.; Franzblau, S.; Möllmann, U. Org. Biol. Chem.2006, 4, 4178-4185. DOI: 10.1039/b612475e
• Syntheses and studies of quinolone-cephalosporins as potential anti-tuberculosis agents. Zhao, G.; Miller, M. J.; Franzblau, S.; Wan, B.; Möllmann, U. Bioorg. Med. Chem. Lett. 2006, 16, 5534-5537. DOI: 10.1016/j.bmcl.2006.08.045
• The Synthesis and in vitro Testing of Structurally Novel Antibiotics Derived from Acylnitroso Diels Alder Adducts. Nora, G. P.; Miller, M. J.; Möllmann, U. Bioorg. Med. Chem. Lett. 2006, 16, 3966-3970. DOI: 10.1016/j.bmcl.2006.05.021
• Stereoselective Total Synthesis of (+)-Streptazolin by Using a Temporary Silicon-tethered RCM Strategy. Li, F.; Miller, M. J. J. Org. Chem. 2006, 71, 5221-5227. DOI: 10.1021/jo060555y
• Substrate Dependent Dihydroxylation of Substituted Cyclopentenes: Towards the Syntheses of Carbocyclic Sinefungin and Noraristeromycin. Jiang, X.; Jin, B.; Gage, J. L.; Miller, M. J. J. Org. Chem. 2006, 71, 4164-4169. DOI: 10.1021/jo060224l
• Molecular Mechanism of Lipopeptide Presentation by CD1a. Zajonc, D. M.; Crispin, M. D. M.; Bowden, T. A.; Young, D. C.; Cheng, T.-Y.; Hu, J.; Costello, C. E.; Rudd, P. M.; Dwek, R. A.; Miller, M. J.; Brenner, M. B.; Moody, D. B.; and Wilson, I. A. Immunity 2005, 22, 209-219. DOI: 10.1016/j.immuni.2004.12.009
• Chemoenzymatic Asymmetric Total Synthesis of Phosphodiesterase Inhibitors: Preparation of a Polycyclic Pyrazolo[3,4- d ]pyrimidine from an Acylnitroso Diels-Alder cycloadduct-Derived Amino Cyclopentenol. Jiang, M.; Warshakoon, N. C.; Miller, M. J. J. Org. Chem. 2005, 70, 2824-2827. DOI: 10.1021/jo0484070
• Desketoneoenactin-Siderophore Conjugates for Candida : Evidence of Iron Transport-Dependent Species Selectivity. Bernier, G.; Girijavallabhan, V.; Murray, A.; Niyaz, N.; Ding, P.; Miller, M. J.; Malouin, F. Antimicrob. Agents Chemother. 2005, 49, 241-248. DOI: 10.1128/AAC.49.1.241-248.2005
• Synthetic Application of Acylnitroso Diels-Alder Derived-Aminocyclopentenols: Total Synthesis of (+)-Streptazolin. Li, F.; Warshakoon, N. C.; Miller, M. J. J.Org. Chem. 2004, 69, 8836-8841. DOI: 10.1021/jo048606j
• Li, F.; Brogan, J. B.; Gage, J. L.; Zhang, D.; Miller, M. J., Chemoenzymatic Synthesis and Synthetic Application of Enantiopure Aminocyclopentenols: Total Synthesis of Carbocyclic (+)-Uracil Polyoxin C and Its a-Epimer. J. Org. Chem. 2004, 69, (13), 4538-4540. DOI: 10.1021/jo0496796
• Lee, W.; Miller, M. J., Concise Synthesis of 4-Acylamino Analogues of 2-Aminobicyclo[ 3.1.0]hexane-2,6-dicarboxylic Acids (LY354740) from an Acylnitroso Diels-Alder Cycloadduct. J. Org. Chem. 2004, 69, (13), 4516-4519. DOI: 10.1021/jo0495034
• Dong, L.; Miller, M. J.; Moellmann, U., Microbial growth promotion studies of exochelin MN and analogues thereof. BioMetals 2004, 17, (2), 99-104. DOI: 10.1023/B:BIOM.0000018348.89904.60
• Ding, P.; Miller, M. J.; Chen, Y.; Helquist, P.; Oliver, A. J.; Wiest, O., Syntheses of Conformationally Constricted Molecules as Potential NAALADase/PSMA Inhibitors. Org. Lett. 2004, 6, (11), 1805-1808. DOI: 10.1021/ol049473r
• Moody, D. B.; Young, D. C.; Cheng, T.-Y.; Rosat, J.-P.; Roura-mir, C.; O'Connor, P. B.; Zajonc, D. M.; Walz, A.; Miller, M. J.; Levery, S. B.; Wilson, I. A.; Costello, C. E.; Brenner, M. B., T Cell Activation by Lipopeptide Antigens. Science 2004, 303, (5657), 527-531. DOI: 10.1126/science.1089353
• Durham, T. B.; Miller, M. J., An Enantioselective Synthesis of Differentially Protected erythro-a,b-Diamino Acids and Its Application to the Synthesis of an Analogue of Rhodopeptin B5. J. Org. Chem. 2003, 68, (1), 35-42. DOI: 10.1021/jo016276m
• Kim, K.-H.; Miller, M. J., An enantioselective synthesis of the cyclopentene fragment of nucleoside Q. Tetrahedron Lett. 2003, 44, (24), 4571-4573. DOI: 10.1016/S0040-4039(03)00973-0
• Oliver, A. J.; Wiest, O.; Helquist, P.; Miller, M. J.; Tenniswood, M., Conformational and SAR analysis of NAALADase and PSMA inhibitors. Bioorg. Med. Chem. 2003, 11, (20), 4455-4461. DOI: 10.1016/S0968-0896(03)00427-9
• Durham, T. B.; Miller, M. J., Enantioselective Synthesis of a-Amino Acids from N-Tosyloxy b-Lactams Derived from b-Keto Esters. J. Org. Chem. 2003, 68, (1), 27-34. DOI: 10.1021/jo0162437
• Dhungana, S.; Miller, M. J.; Dong, L.; Ratledge, C.; Crumbliss, A. L., Iron chelation properties of an extracellular siderophore exochelin MN. J. Am. Chem. Soc. 2003, 125, (25), 7654-7663. DOI: 10.1021/ja029578u
• Lee, W.; Kim, K.-H.; Surman, M. D.; Miller, M. J., Stereo- and Regioselectivity of Pd0/InI-Mediated Allylic Additions to Aldehydes and Ketones. In Situ Generation of Allylindium(III) Intermediates from N-Acylnitroso Diels-Alder Cycloadducts and 1-Amino-4-acetoxycyclopentenes. J. Org. Chem. 2003, 68, (1), 139-149. DOI: 10.1021/jo026488z
• Mineno, T.; Miller, M. J., Stereoselective Total Synthesis of Racemic BCX-1812 (RWJ-270201) for the Development of Neuraminidase Inhibitors as Anti-influenza Agents. J. Org. Chem. 2003, 68, (17), 6591-6596. DOI: 10.1021/jo034316b
• Murray, A. P.; Miller, M. J., The Preparation of a Fully Differentiated "Multiwarhead" Siderophore Precursor. J. Org. Chem. 2003, 68, (1), 191-194. DOI: 10.1021/jo026391c
• Durham, T. B.; Miller, M. J., Conversion of Glucuronic Acid Glycosides to Novel Bicyclic b-Lactams. Org. Lett. 2002, 4, (1), 135-138. DOI: 10.1021/ol017026v
• Surman, M. D.; Mulvihill, M. J.; Miller, M. J., Novel a-substituted b-amino diesters from acylnitroso-derived hetero-Diels-Alder cycloadducts. Tetrahedron Lett. 2002, 43, (7), 1131-1134. DOI: 10.1016/S0040-4039(01)02353-X
• Surman, M. D.; Mulvihill, M. J.; Miller, M. J., Novel 1,4-Benzodiazepines from Acylnitroso-Derived Hetero-Diels-Alder Cycloadducts. Org. Lett. 2002, 4, (1), 139-141. DOI: 10.1021/ol017036w
• Surman, M. D.; Mulvihill, M. J.; Miller, M. J., Regio- and Stereoselective Ring Openings of 3-Aza-2-oxabicyclo[ 2.2.1]hept-5-ene Systems with Copper Catalyst-Modified Grignard Reagents: Application to the Synthesis of an Inhibitor of 5-Lipoxygenase. J. Org. Chem. 2002, 67, (12), 4115-4121. DOI: 10.1021/jo016275u
• Walz, A. J.; Miller, M. J., Synthesis and Biological Activity of Hydroxamic Acid-Derived Vasopeptidase Inhibitor Analogs. Org. Lett. 2002, 4, (12), 2047-2050. DOI: 10.1021/ol025896m
• Dong, L.; Roosenberg, J. M.; Miller, M. J., Total Synthesis of Desferrisalmycin B. J. Am. Chem. Soc. 2002, 124, (50), 15001-15005. DOI: 10.1021/ja028386w
• Dong, L.; Miller, M. J., Total Synthesis of Exochelin MN and Analogues. J. Org. Chem. 2002, 67, (14), 4759-4770. DOI: 10.1021/jo0256078
• Shireman, B. T.; Miller, M. J.; Jonas, M.; Wiest, O., Conformational Study and Enantioselective, Regiospecific Syntheses of Novel Aminoxy trans-Proline Analogues Derived from an Acylnitroso Diels-Alder Cycloaddition. J. Org. Chem. 2001, 66, (18), 6046-6056. DOI: 10.1021/jo010284l
• Lin, Y.-M.; Miller, M. J., Oxidation of Primary Amines to Oxaziridines Using Molecular Oxygen (O2) as the Ultimate Oxidant. J. Org. Chem. 2001, 66, (24), 8282-8285. DOI: 10.1021/jo010965g
• Surman, M. D.; Miller, M. J., Regio- and stereochemically controlled formation of hydroxamic acid containing anti- or syn-1,4-cycloalkenols from acylnitroso-derived Diels-Alder adducts. J. Org. Chem. 2001, 66, (7), 2466-2469. DOI: 10.1021/jo010094a
• Surman, M. D.; Miller, M. J., Synthesis of a Conformationally Restricted Substrate Analogue of Siderophore Biosynthetases. Org. Lett. 2001, 3, (4), 519-521. DOI: 10.1021/ol006813+
• Shireman, B. T.; Miller, M. J., Synthesis of Enantiomerically and Diastereomerically Pure 2(S)-Amino-6(R)-hydroxy-1,7-heptanedioic Acid Dimethyl Ester Hydrochloride from Cycloheptadiene. J. Org. Chem. 2001, 66, (14), 4809-4813. DOI: 10.1021/jo015544d
• Lin, Y.-M.; Miller, M. J.; Mollmann, U., The remarkable hydrophobic effect of a fatty acid side chain on the microbial growth promoting activity of a synthetic siderophore. BioMetals 2001, 14, (2), 153-157. DOI: 10.1023/A:1016666414848
• Vergne, A. F.; Walz, A. J.; Miller, M. J., Iron chelators from mycobacteria (1954-1999) and potential therapeutic applications. Nat. Prod. Rep. 2000, 17, (1), 99-116. DOI: 10.1039/a809397k
• Nurnberger, J. I., Jr.; Adkins, S.; Lahiri, D. K.; Mayeda, A.; Hu, K.; Lewy, A.; Miller, A.; Bowman, E. S.; Miller, M. J.; Rau, N. L.; Smiley, C.; Davis-Singh, D., Melatonin suppression by light in euthymic bipolar and unipolar patients. Arch. Gen. Psychiatry 2000, 57, (6), 572-579. DOI: 10.1001/archpsyc.57.6.572
• Bulychev, A.; Bellettini, J. R.; O'Brien, M.; Crocker, P. J.; Samama, J.-P.; Miller, M. J.; Mobashery, S., N-sulfonyloxy-b-lactam inhibitors for b-lactamases. Tetrahedron 2000, 56, (31), 5719-5728. DOI: 10.1016/S0040-4020(00)00427-0
• Miller, M. J.; Recent Aspects of the Chemistry of b-Lactams--II. Tetrahedron 2000, 56, (31), ix. DOI: 10.1016/S0040-4020(00)00404-X
• Roosenberg, J. M., II; Lin, Y.-M.; Lu, Y.; Miller, M. J., Studies and syntheses of siderophores, microbial iron chelators, and analogs as potential drug delivery agents. Curr. Med. Chem. 2000, 7, (2), 159-197. Link to article
• Li, H.; Miller, M. J., Syntheses and binding studies of oligonucleotides containing N-hydroxycarbamate linkages: potential DNA cleaving antisense oligomers. Tetrahedron Lett. 2000, 41, (22), 4323-4327. DOI: 10.1016/S0040-4039(00)00662-6
• Roosenberg, J. M., II; Miller, M. J., Total Synthesis of the Siderophore Danoxamine. J. Org. Chem. 2000, 65, (16), 4833-4838. DOI: 10.1021/jo000050m

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1990-1999

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• Swaren, P.; Massova, I.; Bellettini, J. R.; Bulychev, A.; Maveyraud, L.; Kotra, L. P.; Miller, M. J.; Mobashery, S.; Samama, J.-P., Elucidation of Mechanism of Inhibition and X-ray Structure of the TEM-1 b-Lactamase from Escherichia coli Inhibited by a N-Sulfonyloxy-b-lactam. Journal of the American Chemical Society 1999, 121, (23), 5353-5359.
• Mourey, L.; Kotra, L. P.; Bellettini, J.; Bulychev, A.; O'Brien, M.; Miller, M. J.; Mobashery, S.; Samama, J.-P., Inhibition of the broad spectrum nonmetallocarbapenamase of class A (NMC-A) b-lactamase from Enterobacter cloacae by monocyclic b-lactams. Journal of Biological Chemistry 1999, 274, (36), 25260-25265.
• Lin, Y.-M.; Miller, M. J., Practical Synthesis of Hydroxamate-Derived Siderophore Components by an Indirect Oxidation Method and Syntheses of a DIG-Siderophore Conjugate and a Biotin-Siderophore Conjugate. Journal of Organic Chemistry 1999, 64, (20), 7451-7458.
• Lu, Y.; Miller, M. J., Syntheses and studies of multiwarhead siderophore-5-fluorouridine conjugates. Bioorganic & Medicinal Chemistry 1999, 7, (12), 3025-3038.
• Li, H.; Miller, M. J., Syntheses of 5'-Deoxy-5'-N-hydroxylaminopyrimidine and Purine Nucleosides: Building Blocks for Novel Antisense Oligonucleosides with Hydroxamate Linkages. Journal of Organic Chemistry 1999, 64, (25), 9289-9293.
• Ghosh, A.; Miller, M. J.; De Clercq, E.; Balzarini, J., Synthesis and biological evaluation of a carbocyclic azanoraristeromycin siderophore conjugate. Nucleosides & Nucleotides 1999, 18, (2), 217-225.
• Lin, Y.-M.; Helquist, P.; Miller, M. J., Synthesis and biological evaluation of a siderophore-Virginiamycin conjugate. Synthesis 1999, (Spec. Iss.), 1510-1514.
• Stocksdale, M. G.; Ramurthy, S.; Miller, M. J., Asymmetric total synthesis of an important 3-(hydroxymethyl)carbacephalosporin. Journal of Organic Chemistry 1998, 63, (4), 1221-1225.
• Vogt, P. F.; Miller, M. J., Development and applications of amino acid-derived chiral acylnitroso hetero Diels-Alder reactions. Tetrahedron 1998, 54, (8), 1317-1348.
• Mulvihill, M. J.; Gage, J. L.; Miller, M. J., Enzymic Resolution of Aminocyclopentenols as Precursors to D- and L-Carbocyclic Nucleosides. Journal of Organic Chemistry 1998, 63, (10), 3357-3363.
• Mulvihill, M. J.; Surman, M. D.; Miller, M. J., Regio- and Stereoselective Fe(III)- and Pd(0)-Mediated Ring Openings of 3-Aza-2-oxabicyclo[ 2.2.1]hept-5-ene Systems. Journal of Organic Chemistry 1998, 63, (15), 4874-4875.
• Mollmann, U.; Ghosh, A.; Dolence, E. K.; Dolence, J. A.; Ghosh, M.; Miller, M. J.; Reissbrodt, R., Selective growth promotion and growth inhibition of Gram-negative and Gram-positive bacteria by synthetic siderophore-b-lactam conjugates. BioMetals 1998, 11, (1), 1-12.
• Mulvihill, M. J.; Miller, M. J., Syntheses of novel hydroxylamine carbanucleosides. Tetrahedron 1998, 54, (24), 6605-6626.
• Zhang, D.; Sueling, C.; Miller, M. J., The Hetero Diels-Alder Reactions between D-Mannose-Derived Halonitroso Compounds and Cyclopentadiene: Scope and Limitations. Journal of Organic Chemistry 1998, 63, (3), 885-888.
• Xu, Y.; Miller, M. J., Total Syntheses of Mycobactin Analogs as Potent Antimycobacterial Agents Using a Minimal Protecting Group Strategy. Journal of Organic Chemistry 1998, 63, (13), 4314-4322.
• Zhang, D.; Miller, M. J., Total Synthesis of (+-) Carbocyclic Polyoxin C and Its a-Epimer. Journal of Organic Chemistry 1998, 63, (3), 755-759.
• Bellettini, J. R.; Miller, M. J., A short synthesis of an important precursor to a new class of bicyclic b-lactamase inhibitors. Tetrahedron Letters 1997, 38, (2), 167-168.
• Vogt, P. F.; Hansel, J.-G.; Miller, M. J., Asymmetric synthesis of an important precursor to 5'-nor carbocyclic nucleosides. Tetrahedron Letters 1997, 38, (16), 2803-2804.
• Miller, M. J.; Darwish, I.; Ghosh, A.; Ghosh, M.; Hansel, J.-G.; Hu, J.; Niu, C.; Ritter, A.; Scheidt, K.; et al., Design, syntheses and studies of new antibacterial, antifungal and antiviral agents. Special Publication - Royal Society of Chemistry 1997, 198, (Anti-Infectives), 116-138.
• Vogt, P. F.; Miller, M. J.; Mulvihill, M. J.; Ramurthy, S.; Savela, G. C.; Ritter, A. R., The synthesis of enantiomerically pure, highly functionalized heterocycles: the products of amino acid based acylnitroso hetero Diels-Alder reactions. Enantiomer 1997, 2, (5), 367-380.
• Hu, J.; Miller, M. J., Total Synthesis of a Mycobactin S, a Siderophore and Growth Promoter of Mycobacterium Smegmatis, and Determination of its Growth Inhibitory Activity against Mycobacterium tuberculosis. Journal of the American Chemical Society 1997, 119, (15), 3462-3468.
• Zhang, D.; Ghosh, A.; Suling, C.; Miller, M. J., Efficient functionalization of acylnitroso cycloadducts: application to the syntheses of carbocyclic nucleoside precursors. Tetrahedron Letters 1996, 37, (22), 3799-3802.
• Niu, C.; Pettersson, T.; Miller, M. J., Enantioselective Total Syntheses of [6R,7R] and [6S,7S] Tricyclic b-Lactams. Journal of Organic Chemistry 1996, 61, (3), 1014-22.
• Ramurthy, S.; Miller, M. J., Framework-reactive siderophore analogs as potential cell-selective drugs. Design and syntheses of trimelamol-based iron chelators. Journal of Organic Chemistry 1996, 61, (12), 4120-4124.
• Diarra, M. S.; Dolence, J. A.; Dolence, E. K.; Darwish, I.; Miller, M. J.; Malouin, F.; Jacques, M., Growth of Actinobacillus pleuropneumoniae is promoted by exogenous hydroxamate and catechol siderophores. Applied and Environmental Microbiology 1996, 62, (3), 853-9.
• Bellettini, J. R.; Miller, M. J., Intermolecular Addition of Amines to an N-Tosyloxy b-Lactam. Journal of Organic Chemistry 1996, 61, (22), 7959-7962.
• Ghosh, A.; Ghosh, M.; Niu, C.; Malouin, F.; Moellmann, U.; Miller, M. J., Iron transport-mediated drug delivery using mixed-ligand siderophore-b-lactam conjugates. Chemistry & Biology 1996, 3, (12), 1011-1019.
• Guzzo, P. R.; Miller, M. J., Nucleophilic addition to the a-carbon of b-lactams. Advances in Nitrogen Heterocycles 1996, 2, 1-34.
• Petty, F.; Rush, A. J.; Davis, J. M.; Calabrese, J. R.; Kimmel, S. E.; Kramer, G. L.; Small, J. G.; Miller, M. J.; Swann, A. E.; et al., Plasma GABA predicts acute response to divalproex in mania. Biological Psychiatry 1996, 39, (4), 278-84.
• Brickman, T. J.; Hansel, J.-G.; Miller, M. J.; Armstrong, S. K., Purification, spectroscopic analysis and biological activity of the macrocyclic dihydroxamate siderophore alcaligin produced by Bordetella pertussis and Bordetella bronchiseptica. BioMetals 1996, 9, (2), 191-203.
• Ghosh, M.; Miller, M. J., Synthesis and in vitro antibacterial activity of spermidine-based mixed catechol- and hydroxamate-containing siderophore-vancomycin conjugates. Bioorganic & Medicinal Chemistry 1996, 4, (1), 43-8.
• Ghosh, M.; Miller, M. J., Synthesis of a bicyclic oxamazin. A novel heteroatom activated b-lactam. Tetrahedron 1996, 52, (12), 4225-38.
• Okonya, J. F.; Kolasa, T.; Miller, M. J., Synthesis of fragments of the peptide component of pseudobactin. Journal of Peptide Science 1996, 2, (3), 157-164.
• Lu, C.; Buyer, J. S.; Okonya, J. F.; Miller, M. J., Synthesis of optically pure chrysobactin and immunoassay development. BioMetals 1996, 9, (4), 377-383.
• Hu, J.; Miller, M. J., An efficient synthesis of cobactin T, a key component of the mycobactin class of siderophores. Tetrahedron Letters 1995, 36, (36), 6379-82.
• Niu, C.; Miller, M. J., Asymmetric syntheses of b-lactams and determination of their absolute configuration. Tetrahedron Letters 1995, 36, (4), 497-500.
• Ghosh, M.; Miller, M. J., Design, synthesis, and biological evaluation of isocyanurate-based antifungal and macrolide antibiotic conjugates: iron transport-mediated drug delivery. Bioorganic & Medicinal Chemistry 1995, 3, (11), 1519-25.
• Hansel, J.-G.; O'Hogan, S.; Lensky, S.; Ritter, A. R.; Miller, M. J., Oxazoline formation via a palladium-catalyzed cyclization: a direct, stereoselective approach to cis-5-amino-2-cyclopenten-1-ol derivatives. Tetrahedron Letters 1995, 36, (17), 2913-16.
• Crocker, P. J.; Miller, M. J., Oxidative free-radical cyclization as a method for annulating b-lactams: syntheses of functionalized carbacephams. Journal of Organic Chemistry 1995, 60, (19), 6176-9.
• Bulychev, A.; O'Brien, M. E.; Massova, I.; Teng, M.; Gibson, T. A.; Miller, M. J.; Mobashery, S., Potent mechanism-based inhibition of the TEM-1 b-lactamase by novel N-sulfonyloxy b-lactams. Journal of the American Chemical Society 1995, 117, (22), 5938-43.
• Crocker, P. J.; Karlsson-Andreasson, U.; Lotz, B. T.; Miller, M. J., Preparation of beta-lactams from beta-hydroxy amides, and annulation of N-malonyl beta-lactams by manganese(III) acetate-promoted free radical cyclization and by aldol cyclization. Heterocycles 1995, 40, (2), 691-716.
• Li, X.; Niu, C.; Miller, M. J., Rearrangement of 3-amido-1-hydroxyazetidin-2-ones. Tetrahedron Letters 1995, 36, (10), 1617-20.
• Ghosh, A.; Ritter, A. R.; Miller, M. J., Synthesis of enantiomerically pure 5'-aza-noraristeromycin analogs. Journal of Organic Chemistry 1995, 60, (18), 5808-13.
• Ghosh, A.; Miller, M. J., Synthesis of novel hydantoin analogs of 5'-nor carbocyclic nucleosides: versatility of a chiral acylnitroso cycloaddition. Tetrahedron Letters 1995, 36, (36), 6399-402.
• Okonya, J. F.; Kolasa, T.; Miller, M. J., Synthesis of the Peptide Fragment of Pseudobactin. Journal of Organic Chemistry 1995, 60, (7), 1932-5.
• Ghosh, M.; Lambert, L. J.; Huber, P. W.; Miller, M. J., Synthesis, bioactivity, and DNA-cleaving ability of desferrioxamine B-nalidixic acid and anthraquinone carboxylic acid conjugates. Bioorganic & Medicinal Chemistry Letters 1995, 5, (20), 2337-40.
• Hu, J.; Miller, M. J., A New Method for the Synthesis ofNe-Acetyl-Ne-hydroxy-L-lysine, the Iron-Binding Constituent of Several Important Siderophores. Journal of Organic Chemistry 1994, 59, (17), 4858-61.
• Ritter, A. R.; Miller, M. J., Amino Acid-Derived Chiral Acyl Nitroso Compounds: Diastereoselectivity in Intermolecular Hetero Diels-Alder Reactions. Journal of Organic Chemistry 1994, 59, (16), 4602-11.
• Ritter, A. R.; Miller, M. J., Asymmetric syntheses of novel amino acids and peptides from acylnitroso-derived cycloadducts. Tetrahedron Letters 1994, 35, (50), 9379-82.
• Guzzo, P. R.; Miller, M. J., Catalytic, Asymmetric Synthesis of the Carbacephem Framework. Journal of Organic Chemistry 1994, 59, (17), 4862-7.
• Ghosh, M.; Miller, M. J., Iron Transport-Mediated Drug Delivery: Synthesis and Biological Evaluation of Cyanuric Acid-Based Siderophore Analogs and b-Lactam Conjugates. Journal of Organic Chemistry 1994, 59, (5), 1020-6.
• Guzzo, P. R.; Miller, M. J., Reactions of N-chloro b-lactams. Tetrahedron 1994, 50, (38), 11091-6.
• Guzzo, P. R.; Teng, M.; Miller, M. J., Synthesis of novel bicyclic b-lactams by intramolecular nucleophile transfer reactions of N-tosyloxy b-lactams. Tetrahedron 1994, 50, (28), 8275-92.
• Darwish, I. S.; Miller, M. J., Synthesis of the Antifungal Agent Neoenactin A and Its N-Deshydroxy Derivative. Journal of Organic Chemistry 1994, 59, (2), 451-4.
• Teng, M.; Miller, M. J.; Nicas, T. I.; Grissom-Arnold, J.; Cooper, R. D. G., b-Lactamase inhibitors derived from N-tosyloxy-b-lactams. Bioorganic & Medicinal Chemistry 1993, 1, (2), 151-4.
• Teng, M.; Gasparski, C. M.; Williams, M. A.; Miller, M. J., A combined electrophilic diazo and nucleophilic azide transfer reaction for the efficient conversion of an N-hydroxy-b-lactam to a carbacephem precursor. Bioorganic & Medicinal Chemistry Letters 1993, 3, (11), 2431-6.
• Stauber, M. J.; Debiak-Krook, T.; Miller, M. J., Alkylation of ambident nucleophilic hydroxamates with 4-substituted 2-azetidinones: formation of bicyclic b-lactam intermediates. Heterocycles 1993, 35, (2), 1205-35.
• Teng, M.; Miller, M. J., Diastereoselective addition of nucleophiles to the C3 position of N-(tosyloxy)-b-lactams. Journal of the American Chemical Society 1993, 115, (2), 548-54.
• Lotz, B. T.; Miller, M. J., Diastereoselective synthesis of the carbacephem framework. Journal of Organic Chemistry 1993, 58, (3), 618-25.
• Ghosh, A.; Miller, M. J., Manganese(III) promoted nitrogen-oxygen bond reduction of N-hydroxy-2-azetidinones. Tetrahedron Letters 1993, 34, (1), 83-6.
• Miller, M. J.; Malouin, F., Microbial iron chelators as drug delivery agents: the rational design and synthesis of siderophore-drug conjugates. Accounts of Chemical Research 1993, 26, (5), 241-9.
• Farouz-Grant, F.; Miller, M. J., Syntheses of novel 1-aminocyclopropane-1-carboxylic acid (ACC)-containing b-lactams. Bioorganic & Medicinal Chemistry Letters 1993, 3, (11), 2423-8.
• Ghosh, A.; Miller, M. J., Synthesis of novel citrate-based siderophores and siderophore-b-lactam conjugates. Iron transport-mediated drug delivery systems. Journal of Organic Chemistry 1993, 58, (27), 7652-9.
• Darwish, I. S.; Patel, C.; Miller, M. J., Synthesis of the antifungal agent norneoenactin A. Journal of Organic Chemistry 1993, 58, (22), 6072-5.
• Gasparski, C. M.; Teng, M.; Miller, M. J., Functionalization of the b-lactam ring: diastereoselective azide transfer and nitrogen-oxygen bond reduction on C4 substituted N-hydroxy-b-lactams in one step. Journal of the American Chemical Society 1992, 114, (7), 2741-3.
• Minnick, A. A.; McKee, J. A.; Dolence, E. K.; Miller, M. J., Iron transport-mediated antibacterial activity of and development of resistance to hydroxamate and catechol siderophore-carbacephalosporin conjugates. Antimicrobial Agents and Chemotherapy 1992, 36, (4), 840-50.
• Gasparski, C. M.; Ghosh, A.; Miller, M. J., Titanium(III)-mediated synthesis of a 1,2,3-tricarbonyl moiety from an a-oximido-b-keto ester: application to the synthesis of the carbacephem nucleus. Journal of Organic Chemistry 1992, 57, (13), 3546-50.
• Ma, C.; Miller, M. J., Asymmetric synthesis of a-hydroxyethyl b-lactam derivatives: an approach to thienamycin. Tetrahedron Letters 1991, 32, (23), 2577-80.
• Minnick, A. A.; Eizember, L. E.; McKee, J. A.; Dolence, E. K.; Miller, M. J., Bioassay for siderophore utilization by Candida albicans. Analytical Biochemistry 1991, 194, (1), 223-9.
• Williams, M. A.; Hsiao, C. N.; Miller, M. J., Direct conversion of N-alkoxy b-lactams to carbapenams: application to the synthesis of the bicyclic PS-5 keto ester. Journal of Organic Chemistry 1991, 56, (8), 2688-94.
• Farouz, F.; Miller, M. J., Facile syntheses and rearrangements of peptide derived b-lactams. Tetrahedron Letters 1991, 32, (28), 3305-8.
• Williams, M. A.; Miller, M. J.; Rath, N. P., Hemiketal formation and subsequent intramolecular acylation of an N-hydroxy b-lactam. Journal of Organic Chemistry 1991, 56, (3), 1293-6.
• McKee, J. A.; Sharma, S. K.; Miller, M. J., Iron transport mediated drug delivery systems: synthesis and antibacterial activity of spermidine- and lysine-based siderophore - b-lactam conjugates. Bioconjugate Chemistry 1991, 2, (4), 281-91.
• Dolence, E. K.; Lin, C. E.; Miller, M. J.; Payne, S. M., Synthesis and siderophore activity of albomycin-like peptides derived from N5-acetyl-N5-hydroxy-L-ornithine. Journal of Medicinal Chemistry 1991, 34, (3), 956-68.
• Dolence, E. K.; Minnick, A. A.; Lin, C. E.; Miller, M. J.; Payne, S. M., Synthesis and siderophore and antibacterial activity of N5-acetyl-N5-hydroxyl-L-ornithine derived siderophore-b-lactam conjugates: iron transport mediated drug delivery. Journal of Medicinal Chemistry 1991, 34, (3), 968-78.
• Gasparski, C. M.; Miller, M. J., Synthesis of b-hydroxy-a-amino acids by aldol condensation using a chiral phase transfer catalyst. Tetrahedron 1991, 47, (29), 5367-78.
• Dolence, E. K.; Miller, M. J., Synthesis of foroxymithine, a microbial fermentation product and angiotensin 1 converting enzyme inhibitor. Journal of Organic Chemistry 1991, 56, (2), 492-9.
• McKee, J. A.; Miller, M. J., Synthesis, siderophore, and antimicrobial evaluation of a spermidine-based tricatecholate siderophore and carbacephalosporin conjugate. Bioorganic & Medicinal Chemistry Letters 1991, 1, (10), 513-18.
• Miller, M. J.; McKee, J. A.; Minnick, A. A.; Dolence, E. K., The design, synthesis and study of siderophore-antibiotic conjugates. Siderophore mediated drug transport. Biology of Metals 1991, 4, (1), 62-9.
• Kolasa, T.; Miller, M. J., 1-Hydroxy-3-amino-2-piperidone (d-N-hydroxycycloornithine) derivatives: key intermediates for the synthesis of hydroxamate-based siderophores. Journal of Organic Chemistry 1990, 55, (6), 1711-21.
• Reno, D. S.; Lotz, B. T.; Miller, M. J., Asymmetric aldol reactions using boron enolates of chiral oxazinones, synthesis of L-allo-threonine. Tetrahedron Letters 1990, 31, (6), 827-30.
• Huang, N. Z.; Kalish, V. J.; Miller, M. J., Double cyclization of aminophosphonoacetate-derived b-hydroxy acids to bicyclic b-lactams. Tetrahedron 1990, 46, (24), 8067-74.
• Dolence, E. K.; Minnick, A. A.; Miller, M. J., N5-Acetyl-N5-hydroxy-L-ornithine-derived siderophore-carbacephalosporin b-lactam conjugates: iron transport mediated drug delivery. Journal of Medicinal Chemistry 1990, 33, (2), 461-4.
• Lotz, B. T.; Gasparski, C. M.; Peterson, K.; Miller, M. J., Substrate specificity studies of aldolase enzymes for use in organic synthesis. Journal of the Chemical Society, Chemical Communications 1990, (16), 1107-9.
• Sheppard, A.; Miller, M. J., Synthesis and reactions of 4-acetoxy-1-oxyazetidin-2-ones. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999) 1990, (9), 2519-25.
• Williams, M. A.; Miller, M. J., Synthesis of the carbapenam ring system via carbene-mediated rearrangement of an N-benzyloxy b-lactam. Tetrahedron Letters 1990, 31, (13), 1807-10.
• Kolasa, T.; Miller, M. J., Synthesis of the chromophore of pseudobactin, a fluorescent siderophore from Pseudomonas. Journal of Organic Chemistry 1990, 55, (14), 4246-55.

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Published before 1990

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• Zercher, C. K.; Miller, M. J., Novel palladium(II)-mediated reactions of N-hydroxy-b-lactams. Tetrahedron Letters 1989, 30, (50), 7009-12.
• Sharma, S. K.; Miller, M. J.; Payne, S. M., Spermexatin and spermexatol: new synthetic spermidine-based siderophore analogs. Journal of Medicinal Chemistry 1989, 32, (2), 357-67.
• Miller, M. J., Syntheses and therapeutic potential of hydroxamic acid based siderophores and analogs. Chemical Reviews ( Washington, DC, United States) 1989, 89, (7), 1563-79.
• Kolasa, T.; Miller, M. J., Syntheses of functionalized b-lactams from tartaric acid. Tetrahedron 1989, 45, (10), 3071-80.
• Hoffman, C.; Tanke, R. S.; Miller, M. J., Synthesis of a-amino acids by reduction of a-oximino esters with titanium(III) chloride and sodium borohydride. Journal of Organic Chemistry 1989, 54, (15), 3750-1.
• Kolasa, T.; Sharma, S. K.; Miller, M. J., a-N-Hydroxy amino acid derivatives. Tetrahedron 1988, 44, (17), 5431-40.
• Kolasa, T.; Miller, M. J., Oxidations of some a-amino acids under Mitsunobu reaction conditions. Tetrahedron Letters 1988, 29, (37), 4661-4.
• Kolasa, T.; Miller, M. J., Studies related to the syntheses of pseudobactin. Pept.: Chem. Biol., Proc. Am. Pept. Symp. 10th 1988, 232-5.
• Huang, N. Z.; Miller, M. J.; Fowler, F. W., Syntheses and flash vacuum pyrolyses of highly functionalized a-N-hydroxy amino acids. Heterocycles 1988, 27, (8), 1821-5.
• Zercher, C. K.; Miller, M. J., Titanium(III) mediated synthesis of dicarboxypyrazines. Heterocycles 1988, 27, (5), 1123-6.
• Rajendra, G.; Miller, M. J., g-Substituent effects on the oxidative cyclization of O-acyl b,g-unsaturated hydroxamates. Tetrahedron Letters 1987, 28, (50), 6257-60.
• Mickel, S. J.; Hsiao, C. N.; Miller, M. J., 4-Acetoxyazetidin-2-one: synthesis of a key beta-lactam intermediate by a [2 + 2] cycloaddition route [2-azetidinone, 4-(acetyloxy)-]. Organic Syntheses 1987, 65, 135-9.
• Hsiao, C. N.; Liu, L.; Miller, M. J., Cysteine- and serine-derived thiazolidinethiones and oxazolidinethiones as efficient chiral auxiliaries in aldol condensations. Journal of Organic Chemistry 1987, 52, (11), 2201-6.
• Boyd, D. B.; Eigenbrot, C.; Indelicato, J. M.; Miller, M. J.; Pasini, C. E.; Woulfe, S. R., Heteroatom-activated b-lactam antibiotics: considerations of differences in the biological activity of [[3(S)-(acylamino)-2-oxo-1-azetidinyl]oxy]acetic acids (oxamazins) and the corresponding sulfur analogs (thiamazins). Journal of Medicinal Chemistry 1987, 30, (3), 528-36.
• Rajendra, G.; Miller, M. J., Intramolecular electrophilic additions to olefins in organic syntheses. Stereoselective synthesis of 3,4-substituted b-lactams by bromine-induced oxidative cyclization of O-acyl b,g-unsaturated hydroxamic acid derivatives. Journal of Organic Chemistry 1987, 52, (20), 4471-7.
• Kolasa, T.; Miller, M. J., Reactions of a-hydroxy carbonyl compounds with azodicarboxylates and triphenylphosphine: synthesis of a-N-hydroxy amino acid derivatives. Journal of Organic Chemistry 1987, 52, (22), 4978-84.
• Kolasa, T.; Sharma, S.; Miller, M. J., Reactions of organometallics with oximes. Synthesis of N-hydroxy a-amino acids. Tetrahedron Letters 1987, 28, (42), 4973-6.
• Biswas, A.; Miller, M. J., Rearrangement of N-(p-toluenesulfonyloxy)-2-pyrrolidinone. Heterocycles 1987, 26, (11), 2849-51.
• Kolasa, T.; Miller, M. J., Synthesis of substituted 3-hydroxy-4-(alkoxycarbonyl)-2-azetidinones. Tetrahedron Letters 1987, 28, (17), 1861-4.
• Lee, B. H.; Biswas, A.; Miller, M. J., [1,2]-Anionic rearrangements of substituted N-hydroxy-2-azetidinones and applications to the synthesis of bicyclic b-lactams. Journal of Organic Chemistry 1986, 51, (1), 106-9.
• Kolasa, T.; Miller, M. J., A simple method for distinguishing optical isomers of chiral amines, hydroxylamines, amino acids, and peptides. Journal of Organic Chemistry 1986, 51, (15), 3055-8.
• Liu, L.; Tanke, R. S.; Miller, M. J., Electrophilic sulfur transfer reactions in organic synthesis. Preparation of a diastereomer of the key macrocyclic component of griseoviridin. Journal of Organic Chemistry 1986, 51, (26), 5332-7.
• Miller, M. J., Hydroxamate approach to the synthesis of b-lactam antibiotics. Accounts of Chemical Research 1986, 19, (2), 49-56.
• Iwagami, H.; Woulfe, S. R.; Miller, M. J., Reactions of [(2-oxo-1-azetidinyl)thio]phthalimides with nucleophiles. Tetrahedron Letters 1986, 27, (27), 3095-8.
• Biswas, A.; Eigenbrot, C.; Miller, M. J., Rearrangements of N-hydroxy b-lactams. Tetrahedron 1986, 42, (23), 6421-8.
• Woulfe, S. R.; Miller, M. J., The synthesis of substituted [[3(S)-(acylamino)-2-oxo-1-azetidinyl]thio]acetic acids. Journal of Organic Chemistry 1986, 51, (16), 3133-9.
• Krook, M. A.; Miller, M. J.; Eigenbrot, C., A novel rearrangement of 3-phenylacetamido-1-hydroxyazetidin-2-one. Journal of the Chemical Society, Chemical Communications 1985, (18), 1265-6.
• Lee, B. H.; Miller, M. J.; Prody, C. A.; Neilands, J. B., Artificial siderophores. 1. Synthesis and microbial iron transport capabilities. Journal of Medicinal Chemistry 1985, 28, (3), 317-23.
• Lee, B. H.; Miller, M. J.; Prody, C. A.; Neilands, J. B., Artificial siderophores. 2. Syntheses of trihydroxamate analogs of rhodotorulic acid and their biological iron transport capabilities in Escherichia coli. Journal of Medicinal Chemistry 1985, 28, (3), 323-7.
• Woulfe, S. R.; Iwagami, H.; Miller, M. J., Efficient N-sulfenylation of 2-azetidinones using S-substituted thiophthalimides. Tetrahedron Letters 1985, 26, (33), 3891-4.
• Hsiao, C. N.; Ashburn, S. P.; Miller, M. J., Enantioselective aldol reaction of chiral acylthiazolidinethione-derived boron enolates. Tetrahedron Letters 1985, 26, (40), 4855-8.
• Rajendra, G.; Miller, M. J., Oxidative cyclization of b,g-unsaturated O-acyl hydroxamates to b-lactams. Tetrahedron Letters 1985, 26, (44), 5385-8.
• Woulfe, S. R.; Miller, M. J., Synthesis and biological activity of substituted [[3(S)-(acylamino)-2-oxo-1-azetidinyl]oxy]acetic acids. A new class of heteroatom-activated b-lactam antibiotics. Journal of Medicinal Chemistry 1985, 28, (10), 1447-53.
• Jung, M.; Miller, M. J., The application of highly stereoselective aldol condensations to the synthesis of b-lactam antibiotics. Tetrahedron Letters 1985, 26, (8), 977-80.
• Krook, M. A.; Miller, M. J., The direct cyclization of a-acylamino-substituted hydroxamates to b-lactams. Journal of Organic Chemistry 1985, 50, (7), 1126-8.
• Lee, B. H.; Gerfen, G. J.; Miller, M. J., Constituents of microbial iron chelators. Alternate syntheses of d-N-hydroxy-L-ornithine derivatives and applications to the synthesis of rhodotorulic acid. Journal of Organic Chemistry 1984, 49, (13), 2418-23.
• Lee, B. H.; Miller, M. J., Constituents of microbial iron chelators. The synthesis of optically active derivatives of d-N-hydroxy-L-ornithine. Tetrahedron Letters 1984, 25, (9), 927-30.
• Woulfe, S. R.; Miller, M. J., Heteroatom activated b-lactam antibiotics: synthesis of biologically active substituted N-oxy-3-amino-2-azetidinones (oxamazins). Tetrahedron Letters 1984, 25, (31), 3293-6.
• Mattingly, P. G.; Miller, M. J.; Cooper, R. D. G.; Daughtery, B. W., Chiral synthesis of protected 3-amino-4-(alkoxycarbonyl)-2-azetidinones from b-hydroxyaspartic acid. Journal of Organic Chemistry 1983, 48, (20), 3556-9.
• Morrison, M. A.; Miller, M. J., Conversion of b-hydroxyglutarohydroxamates to carbapenem precursors. Journal of Organic Chemistry 1983, 48, (23), 4421-3.
• Capecchi, J. T.; Miller, M. J.; Loudon, G. M., Critical examination of a method for the analysis of a and w linkages in peptides containing aspartic acid and glutamic acid. Journal of Organic Chemistry 1983, 48, (12), 2014-21.
• Lee, B. H.; Miller, M. J., Natural ferric ionophores: total synthesis of schizokinen, schizokinen A, and arthrobactin. Journal of Organic Chemistry 1983, 48, (1), 24-31.
• Miller, M. J.; Biswas, A.; Krook, M. A., Practical synthetic approaches to intermediates for the preparation of the novel O-sulfonated-N-hydroxy-2-azetidinone antibiotics. Tetrahedron 1983, 39, (15), 2571-5.
• Bajwa, J. S.; Miller, M. J., Preparation of chiral substituted succinic acids. Journal of Organic Chemistry 1983, 48, (7), 1114-16.
• Maurer, P. J.; Miller, M. J., Total synthesis of a mycobactin: mycobactin S2. Journal of the American Chemical Society 1983, 105, (2), 240-5.
• Miller, M. J.; Bajwa, J. S.; Mattingly, P. G.; Peterson, K., Enantioselective syntheses of 3-substituted 4-(alkoxycarbonyl)-2-azetidinones from malic acid. Journal of Organic Chemistry 1982, 47, (25), 4928-33.
• Maurer, P. J.; Miller, M. J., Microbial iron chelators: total synthesis of aerobactin and its constituent amino acid, N6-acetyl-N6-hydroxylysine. Journal of the American Chemical Society 1982, 104, (11), 3096-101.
• Maurer, P. J.; Miller, M. J., Mycobactins: synthesis of (-)-cobactin T from e-hydroxynorleucine. Journal of Organic Chemistry 1981, 46, (13), 2835-6.
• Mattingly, P. G.; Miller, M. J., Synthesis of 2-azetidinones from serinehydroxamates: approaches to the synthesis of 3-aminonocardicinic acid. Journal of Organic Chemistry 1981, 46, (8), 1557-64.
• Miller, M. J., Isourea-mediated preparation of dehydro amino acids. Journal of Organic Chemistry 1980, 45, (15), 3131-2.
• Miller, M. J.; Mattingly, P. G.; Morrison, M. A.; Kerwin, J. F., Jr., Synthesis of b-lactams from substituted hydroxamic acids. Journal of the American Chemical Society 1980, 102, (23), 7026-32.
• Mattingly, P. G.; Miller, M. J., Titanium trichloride reduction of substituted N-hydroxy-2-azetidinones and other hydroxamic acids. Journal of Organic Chemistry 1980, 45, (3), 410-15.
• Mattingly, P. G.; Kerwin, J. F., Jr.; Miller, M. J., A facile synthesis of substituted N-hydroxy-2-azetidinones. A biogenetic type b-lactam synthesis. Journal of the American Chemical Society 1979, 101, (14), 3983-5.

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2000 to present

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• (WO/2009/158118) ANTI-BACTERIAL AGENTS FROM BENZO[D]HETEROCYCLIC SCAFFOLDS FOR PREVENTION AND TREATMENT OF MULTIDRUG RESISTANT BACTERIA

  Applicants:

  UNIVERSITY OF NOTRE DAME DU LAC [US/US]; 511 Main Building Notre Dame, IN 46556-5602 (US)(All Except US). MILLER, Marvin, J. [US/US]; (US) (US Only). MORASKI, Garrett, C. [US/US]; (US) (US Only).

• (WO/2009/111502) ANTI-CANCER COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME

  Applicants:

  UNIVERSITY OF NOTRE DAME DU LAC [US/US]; 511 Main Building Notre Dame, IN 46556-5602 (US)(All Except US). MILLER, Marvin, J. [US/US]; (US) (US Only). MORASKI, Garrett, C. [US/US]; (US) (US Only). STEFELY, Jonathan [US/US]; (US) (US Only).

• “Beta.-Lactamyl vasopressin V.sub.1a Antagonists.” Bruns, Jr.; Robert F. (Carmel, IN) , Guillon; Christophe D. G. (Bethlehem, PA) , Heindel; Ned D. (Easton, PA) , Koppel; Gary A. (Indianapolis, IN) , Miller; Marvin J. (South Bend, IN), US Patent 7,119,083, October 10, 2006.
• Bruns, R. F., Jr.; Guillon, C. D. G.; Heindel, N. D.; Koppel, G. A.; Lu, S.; Miller, M. J.; Simon, N. G. Preparation of peptidyl b-lactams as vasopressin V 1a antagonists. PCT Int. Appl. 2003031407, 2003.
• "Cyclopentenyl Hydroxamic Acid-Derived Inhibitor of 5-Lipoxygenase." Marvin J. Miller and Matthew D. Surman, Provisional Patent Pending, filed January 4, 2002.
• "Hydroxamic Acid-Derived Vasopeptidase Inhibitors." Marvin J. Miller and Andrew Walz, Provisional Patent Pending, filed January 4, 2002.
• "Heterocyclic Antituberculosis." Marvin J. Miller and Jingdan Hu , US Patent 6,403,623 B1, (provisional), June 11, 2002.
• "Antimycobacterial Agents." Marvin J. Miller, Yanping Xu, US Patent 6,310,058 B1 (provisional), October 30, 2001.

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Issued before 2000

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• “Antibacterial and Antifungal Nucleosides.” Marvin J. Miller, Julia M. Dolence, Manuka Ghosh, US Patent 5,783,689, July 21, 1998.
• “Bicyclic Beta-Lactams and Process Therefor.” Min Teng and Marvin J. Miller, US Patent 5,750,681, May 12, 1998.
• "Process for the Preparation of 3-Substituted-2-Azetidinones." Marvin J. Miller, Catherine M. Gasparski, C. M., Min Teng, US Patent 5,250, 676, October 5, 1993.
• "Beta-Hydroxy-Alpha-Amino Acids." Marvin J. Miller, U.S. Patent 5,266,468, November 30, 1993; South Africa 91/4201; February 24, 1993; New Zealand 238342.
• "Process for Bicyclic b -Lactams Diazo- b -keto-butyrate-intermediates for Bicyclic ß-Lactams." Marvin J. Miller and Matthew A. Williams, US Patent 5,106,968, April 21, 1992.
• "Rhodium Catalyzed Cyclization Process for Bicyclic b -Lactams." Marvin J. Miller and Matthew A. Williams, US Patent 5,051,502, September 24, 1991; Taiwan N158455, January 12, 1993.
• "Monocyclic Beta-Lactams and Processes for the Preparation Thereof." Marvin J. Miller, US Patent 4,992,544, February 12, 1991.
• "Process for Intermediates to 1-Carbapenems and 1-Carbacephems." Chi-nung W. Hsiao and Marvin J. Miller, US Patent 4,845,229, July 4, 1989; Israel 94673, September 19, 1992.
• "Azetidinone N-Phosphonomethyl Esters." Marvin J. Miller, US Patent 4,820,815, April 11, 1989.
• "Process for 4-Halomethyl-azetidinones by Cyclization of O-Azetidinones." Marvin J. Miller, US Patent 4,751,296, June 14, 1988; Taiwan N133442, December 4, 1989; Israel 83420, October 16, 1992; Hungary 201737, August 15, 1990; European Patent Office 0256763, December 8, 1993; Canada 1282066, March 26, 1991.
• "Process for Intermediates to 1-Carbapenems and 1-Carbapenams." C.-N. W. Hsiao and Marvin J. Miller, US Patent 4,745,201, May 17, 1988; United Kingdom 0218415, August 8, 1990; Taiwan N134225, January 23, 1990; Switzerland 0218415, August 8, 1990; Sweden 0218415, August 8, 1990; Netherlands 0218415, August 8, 1990; Korea 25766, July 28, 1988; Italy 0218415, August 8, 1990; Israel 80128, May 17, 1992; Hungary 198464, June 27, 18989; West Germany P3673306.7-08, August 8, 1990; France 0218415, August 8, 1990; European Patent Office 0218415, August 8, 1990; Canada 1304744, July 7, 1992; Belgium 0218415, August 8, 1990; Austria E55383, August 8, 1990.
• "Cyclization Process for b -Lactams." Marvin J. Miller, US Patent 4,675,399, June 23, 1987.
• "N-(Substituted-Methyl)-Azetidin-2-ones." Marvin J. Miller, US Patent 4,595,532, June 17, 1986; United Kingdom 2134902, April 1, 1987; Korea 23285, May 11, 1987; Hungary 195772, April 29, 1988; Greece 81665, December 12, 1984; Canada 1267415, April 3, 1990.

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